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The responsible enzyme can be blocked by entacapone, allowing higher levels of L-dopa and dopamine to be achieved in corpus striatum. Anticholinergics. Antagonists at muscarinic cholinoceptors, such as benzatropine and biperiden (p. 106), suppress striatal cholinergic overactivity and thereby relieve rigidity and tremor; however, akinesia is not reversed or is even exacerbated.
Hence, pirenzepine may act by blocking M1 receptors on ECL cells or submucosal neurons. Histamine receptors on parietal cells belong to the H2 type and are blocked by H2-antihistamines. |
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